40 complex(es)
PDB ID
Protein Name
Organism
Uniprot ID/ACC
Ligand Name
HET ID
Structure
PS-Score (Pocket Similarity)
Card
1 6G29 Histone-lysine N-methyltransferase NSD3 Homo sapiens Q9BZ95 (NSD3_HUMAN) 5-methyl-2-piperidin-4-yl-6-pyridin-4-yl-pyridazin-3-one EHK 0.95 SHOW
2 6G2C Histone-lysine N-methyltransferase NSD3 Homo sapiens Q9BZ95 (NSD3_HUMAN) 3,5-dimethyl-4-(1-methyl-5-pyridin-4-yl-imidazol-4-yl)-1,2-oxazole EHT 0.9 SHOW
3 6G2E Histone-lysine N-methyltransferase NSD3 Homo sapiens Q9BZ95 (NSD3_HUMAN) [3,5-dimethyl-4-(1-methyl-5-pyridin-4-yl-imidazol-4-yl)phenyl]methanamine EHH 0.88 SHOW
4 6G2F Histone-lysine N-methyltransferase NSD3 Homo sapiens Q9BZ95 (NSD3_HUMAN) 4-[5-(7-fluoranylquinolin-4-yl)-1-methyl-imidazol-4-yl]-3,5-dimethyl-1,2-oxazole EHW 0.84 SHOW
5 6G2O Histone-lysine N-methyltransferase NSD3 Homo sapiens Q9BZ95 (NSD3_HUMAN) [4-[5-(7-fluoranylquinolin-4-yl)-1-methyl-imidazol-4-yl]-3,5-dimethyl-phenyl]methanamine EJE 0.83 SHOW
6 6G2B Histone-lysine N-methyltransferase NSD3 Homo sapiens Q9BZ95 (NSD3_HUMAN) 4-(3-methyl-5-phenyl-imidazol-4-yl)pyridine EH8 0.77 SHOW
7 6G25 Histone-lysine N-methyltransferase NSD3 Homo sapiens Q9BZ95 (NSD3_HUMAN) 3,5-dimethyl-4-(4-pyridin-4-yl-1~{H}-pyrazol-3-yl)-1,2-oxazole EHQ 0.74 SHOW
8 3MO8 Peregrin Homo sapiens P55201 (BRPF1_HUMAN) N-TRIMETHYLLYSINE M3L 0.73 SHOW
9 3QJ6 Hepatoma-derived growth factor-related protein 2 Homo sapiens Q7Z4V5 (HDGR2_HUMAN) N-TRIMETHYLLYSINE M3L 0.73 SHOW
10 5C6S Peregrin Homo sapiens P55201 (BRPF1_HUMAN) isoquinoline-3-carboxylic acid 4K8 0.6 SHOW
11 5NRV DNA (cytosine-5)-methyltransferase 3B Homo sapiens Q9UBC3 (DNM3B_HUMAN) 6-dipropylamino-1-hexanol 96K 0.6 SHOW
12 6KCU JIL-1 anchoring and stabilizing protein, isoform A Drosophila melanogaster Q9VAA9 (Q9VAA9_DROME) 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL BTB 0.59 SHOW
13 2X4Y Peregrin Homo sapiens P55201 (BRPF1_HUMAN) N-TRIMETHYLLYSINE M3L 0.59 SHOW
14 6IIS Hepatoma-derived growth factor-related protein 3 Homo sapiens Q9Y3E1 (HDGR3_HUMAN) N-TRIMETHYLLYSINE M3L 0.57 SHOW
15 4N4H Zinc finger MYND domain-containing protein 11 Mus musculus Q8R5C8 (ZMY11_MOUSE) N-TRIMETHYLLYSINE M3L 0.57 SHOW
16 6IIT Hepatoma-derived growth factor-related protein 3 Homo sapiens Q9Y3E1 (HDGR3_HUMAN) N-DIMETHYL-LYSINE MLY 0.57 SHOW
17 3QBY Hepatoma-derived growth factor-related protein 2 Homo sapiens Q7Z4V5 (HDGR2_HUMAN) N-TRIMETHYLLYSINE M3L 0.57 SHOW
18 4N4I Zinc finger MYND domain-containing protein 11 Mus musculus Q8R5C8 (ZMY11_MOUSE) N-TRIMETHYLLYSINE M3L 0.56 SHOW
19 5NRR DNA (cytosine-5)-methyltransferase 3B Homo sapiens Q9UBC3 (DNM3B_HUMAN) 5-[2-hydroxyethyl(propyl)amino]pentan-1-ol 96E 0.55 SHOW
20 5CIU DNA (cytosine-5)-methyltransferase 3B Homo sapiens Q9UBC3 (DNM3B_HUMAN) N-TRIMETHYLLYSINE M3L 0.54 SHOW
21 6G3T Histone-lysine N-methyltransferase NSD3 Homo sapiens Q9BZ95 (NSD3_HUMAN) 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID EPE 0.54 SHOW
22 2X4X Peregrin Homo sapiens P55201 (BRPF1_HUMAN) N-TRIMETHYLLYSINE M3L 0.53 SHOW
23 3QKJ DNA (cytosine-5)-methyltransferase 3B Homo sapiens Q9UBC3 (DNM3B_HUMAN) 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL BTB 0.53 SHOW
24 5NRS DNA (cytosine-5)-methyltransferase 3B Homo sapiens Q9UBC3 (DNM3B_HUMAN) (2~{S})-1-[2-hydroxyethyl-[(2~{S})-2-oxidanylpropyl]amino]propan-2-ol 962 0.53 SHOW
25 2X4W Peregrin Homo sapiens P55201 (BRPF1_HUMAN) N-TRIMETHYLLYSINE M3L 0.52 SHOW
26 5NV0 DNA (cytosine-5)-methyltransferase 3B Homo sapiens Q9UBC3 (DNM3B_HUMAN) 4-(dipropylamino)butanenitrile 9AH 0.52 SHOW
27 6R3E DNA (cytosine-5)-methyltransferase 3B Homo sapiens Q9UBC3 (DNM3B_HUMAN) Triisopropanolamine 96H 0.51 SHOW
28 5NR3 DNA (cytosine-5)-methyltransferase 3B Homo sapiens Q9UBC3 (DNM3B_HUMAN) Ethambutol 95E 0.49 SHOW
29 5VAR Lysine-specific demethylase 4A Homo sapiens O75164 (KDM4A_HUMAN) (1R,2S,3R,4S)-3-[(dimethylamino)methyl]-1-phenylbicyclo[2.2.1]heptan-2-ol 92Y 0.48 SHOW
30 5NV2 DNA (cytosine-5)-methyltransferase 3B Homo sapiens Q9UBC3 (DNM3B_HUMAN) (2~{S})-6-methyl-~{N}-propan-2-yl-heptan-2-amine 9AE 0.47 SHOW
31 6BHD Histone-lysine N-methyltransferase SETDB1 Homo sapiens Q15047 (SETB1_HUMAN) N-DIMETHYL-LYSINE MLY 0.47 SHOW
32 5D6Y Lysine-specific demethylase 4A Homo sapiens O75164 (KDM4A_HUMAN) N-TRIMETHYLLYSINE M3L 0.44 SHOW
33 2GFA Lysine-specific demethylase 4A Homo sapiens O75164 (KDM4A_HUMAN) N-TRIMETHYLLYSINE M3L 0.43 SHOW
34 4BD3 PHD finger protein 19 Homo sapiens Q5T6S3 (PHF19_HUMAN) N-TRIMETHYLLYSINE M3L 0.42 SHOW
35 6X47 Gag-Pol polyprotein Human immunodeficiency virus type 1 group M subtype B P03366 (POL_HV1B1) 7-(2-(2-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)ethoxy)phenoxy)-2-naphthonitrile 7AX 0.42 SHOW
36 6BHE Histone-lysine N-methyltransferase SETDB1 Homo sapiens Q15047 (SETB1_HUMAN) N-TRIMETHYLLYSINE M3L 0.42 SHOW
37 5NV7 DNA (cytosine-5)-methyltransferase 3B Homo sapiens Q9UBC3 (DNM3B_HUMAN) N1-(2-hydroxyethyl)-2-methyl-1,2-propanediamine 9AK 0.42 SHOW
38 3MEU SAGA-associated factor 29 Homo sapiens Q96ES7 (SGF29_HUMAN) N-TRIMETHYLLYSINE M3L 0.42 SHOW
39 2R58 Polycomb protein Scm Drosophila melanogaster Q9VHA0 (SCM_DROME) N-DIMETHYL-LYSINE MLY 0.41 SHOW
40 3MP1 SAGA-associated factor 29 Saccharomyces cerevisiae P25554 (SGF29_YEAST) N-TRIMETHYLLYSINE M3L 0.41 SHOW