Protein Download |
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Protein Name | Lysine-specific demethylase 4A | |
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#PDB ID | 16 | |
Organism | Homo sapiens | |
Uniprot ID/ACC | O75164 (KDM4A_HUMAN) | |
Protein Sequence | MASESETLNPSARIMTFYPTMEEFRNFSRYIAYIESQGAHRAGLAKVVPPKEWKPRASYDDIDDLVIPAPIQQLVTGQSGLFTQYNIQKKAMTVREFRKIANSDKYCTPRYSEFEELERKYWKNLTFNPPIYGADVNGTLYEKHVDEWNIGRLRTILDLVEKESGITIEGVNTPYLYFGMWKTSFAWHTEDMDLYSINYLHFGEPKSWYSVPPEHGKRLERLAKGFFPGSAQSCEAFLRHKMTLISPLMLKKYGIPFDKVTQEAGEFMITFPYGYHAGFNHGFNCAESTNFATRRWIEYGKQAVLCSCRKDMVKISMDVFVRKFQPERYKLWKAGKDNTVIDHTLPTPEAAEFLKESELPPRAGNEEECPEEDMEGVEDGEEGDLKTSLAKHRIGTKRHRVCLEIPQEVSQSELFPKEDLSSEQYEMTECPAALAPVRPTHSSVRQVEDGLTFPDYSDSTEVKFEELKNVKLEEEDEEEEQAAAALDLSVNPASVGGRLVFSGSKKKSSSSLGSGSSRDSISSDSETSEPLSCRAQGQTGVLTVHSYAKGDGRVTVGEPCTRKKGSAARSFSERELAEVADEYMFSLEENKKSKGRRQPLSKLPRHHPLVLQECVSDDETSEQLTPEEEAEETEAWAKPLSQLWQNRPPNFEAEKEFNETMAQQAPHCAVCMIFQTYHQVEFGGFNQNCGNASDLAPQKQRTKPLIPEMCFTSTGCSTDINLSTPYLEEDGTSILVSCKKCSVRVHASCYGVPPAKASEDWMCSRCSANALEEDCCLCSLRGGALQRANDDRWVHVSCAVAILEARFVNIAERSPVDVSKIPLPRFKLKCIFCKKRRKRTAGCCVQCSHGRCPTAFHVSCAQAAGVMMQPDDWPFVVFITCFRHKIPNLERAKGALQSITAGQKVISKHKNGRFYQCEVVRLTTETFYEVNFDDGSFSDNLYPEDIVSQDCLQFGPPAEGEVVQVRWTDGQVYGAKFVASHPIQMYQVEFEDGSQLVVKRDDVYTLDEELPKRVKSRLSVASDMRFNEIFTEKEVKQEKKRQRVINSRYREDYIEPALYRAIME | |
Protein Class | TRANSCRIPTION REGULATOR | |
Synonym(s) |
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Gene Symbol | KDM4A | |
Gene ID | 9682 | |
Pfam ID | PF02373, PF02375, PF18104 | |
Interpro ID | IPR034732, IPR003347, IPR003349, IPR040477, IPR002999, IPR011011, IPR001965, IPR013083 |
Bound Ligands |
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HET ID | Ligand Type | PDB ID | Binding Affinity | Binding Database | Structure | Complex Card |
FQE | Small Molecule | 6H4S | Ki : 2.0 nM | Binding MOAD | |
SHOW |
FQB | Small Molecule | 6H4R | Ki : 0.004 nM | Binding MOAD | |
SHOW |
FOW | Small Molecule | 6H4T | Ki : 4.0 nM | Binding MOAD | |
SHOW |
FQN | Small Molecule | 6H4V | IC50 : 613.0 nM | Binding MOAD | |
SHOW |
FO8 | Small Molecule | 6H4Y | IC50 : 77.0 nM | Binding MOAD | |
SHOW |
FNQ | Small Molecule | 6H4X | IC50 : 131.0 nM | Binding MOAD | |
SHOW |
FQH | Small Molecule | 6H4O | IC50 : 128.0 nM | Binding MOAD | |
SHOW |
FQ5 | Small Molecule | 6H4P | Ki : 3.0 nM | Binding MOAD | |
SHOW |
92Y | Small Molecule | 5VAR | Kd : 81700.0 nM | Binding MOAD | |
SHOW |
OGA | Small Molecule | 5LY2 |
- |
- |
|
SHOW |
M3L | H3K23me3 | 5D6Y |
- |
- |
|
SHOW |
M3L | H4K20me3 | 2QQS |
- |
- |
|
SHOW |
FO2 | Small Molecule | 6H4U |
- |
- |
|
SHOW |
QC1 | Small Molecule | 6CG1 |
- |
- |
|
SHOW |
M3L | H3K4me3 | 2GFA |
- |
- |
|
SHOW |
FQQ | Small Molecule | 6H4W |
- |
- |
|
SHOW |