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Protein Download |
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| Protein Name | Choline kinase alpha | |||||
|---|---|---|---|---|---|---|
| #PDB ID | 14 | |||||
| Organism | Homo sapiens | |||||
| Uniprot ID/ACC | P35790 (CHKA_HUMAN) | |||||
| Protein Sequence | MKTKFCTGGEAEPSPLGLLLSCGSGSAAPAPGVGQQRDAASDLESKQLGGQQPPLALPPPPPLPLPLPLPQPPPPQPPADEQPEPRTRRRAYLWCKEFLPGAWRGLREDEFHISVIRGGLSNMLFQCSLPDTTATLGDEPRKVLLRLYGAILQMRSCNKEGSEQAQKENEFQGAEAMVLESVMFAILAERSLGPKLYGIFPQGRLEQFIPSRRLDTEELSLPDISAEIAEKMATFHGMKMPFNKEPKWLFGTMEKYLKEVLRIKFTEESRIKKLHKLLSYNLPLELENLRSLLESTPSPVVFCHNDCQEGNILLLEGRENSEKQKLMLIDFEYSSYNYRGFDIGNHFCEWMYDYSYEKYPFFRANIRKYPTKKQQLHFISSYLPAFQNDFENLSTEEKSIIKEEMLLEVNRFALASHFLWGLWSIVQAKISSIEFGYMDYAQARFDAYFHQKRKLGV | |||||
| Protein Class | TRANSFERASE | |||||
| Synonym(s) |
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| Gene Symbol | CHKA | |||||
| Gene ID | 1119 | |||||
| Pfam ID | - | |||||
| Interpro ID | IPR011009 |
Bound Ligands |
HET ID | Ligand Type | PDB ID | Binding Affinity | Binding Database | Structure | Complex Card |
| U85 | Small Molecule | 4BR3 | Kd : 1900.0 nM | PDBBind | |
SHOW |
| U85 | Small Molecule | 4BR3 | Kd : 1900.0 nM | Binding MOAD | |
SHOW |
| HC6 | Small Molecule | 3G15 | Kd : 100.0 nM | PDBBind | |
SHOW |
| 0H7 | Small Molecule | 4DA5 | Ki : 360.0 nM | PDBBind | |
SHOW |
| 0H7 | Small Molecule | 4DA5 | Ki : 360.0 nM | Binding MOAD | |
SHOW |
| 5RA | Small Molecule | 5EQY | Kd : 10.0 nM, Kd : 66.0 nM | BindingDB | |
SHOW |
| 5RA | Small Molecule | 5EQY | IC50 : 70.0 nM | Binding MOAD | |
SHOW |
| 5R8 | Small Molecule | 5EQE | Kd : 132000.0 nM, Kd : 87000.0 nM | BindingDB | |
SHOW |
| 5R8 | Small Molecule | 5EQE | IC50 : 87000.0 nM | Binding MOAD | |
SHOW |
| 5R9 | Small Molecule | 5EQP | Kd : 4000.0 nM, Kd : 3900.0 nM | BindingDB | |
SHOW |
| 5R9 | Small Molecule | 5EQP | IC50 : 3900.0 nM | Binding MOAD | |
SHOW |
| G8S | Small Molecule | 4CG8 | IC50 : 1200.0 nM | Binding MOAD | |
SHOW |
| NBR | Small Molecule | 5FTG | Kd : 700.0 nM | Binding MOAD | |
SHOW |
| QTH | Small Molecule | 7A06 |
- |
- |
|
SHOW |
| HC6 | Small Molecule | 3F2R |
- |
- |
|
SHOW |
| QLW | Small Molecule | 4CGA |
- |
- |
|
SHOW |
| QTK | Small Molecule | 7A04 |
- |
- |
|
SHOW |
| GQG | Small Molecule | 4CG9 |
- |
- |
|
SHOW |
| PC | Small Molecule | 2CKQ |
- |
- |
|
SHOW |